TOPIC

Anabolic Steroids

Anabolic SteroidsSparse/variable compound-specific evidence

Mestanolone

Mestanolone is listed in current U.S. federal Schedule III regulations as an anabolic steroid or covered anabolic-steroid substance. Compound-specific human evidence may be limited or historical.

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Anabolic SteroidsSparse/variable compound-specific evidence

Epithio-17α-methyl-androstanol

Epithio-17α-methyl-androstanol is listed in current U.S. federal Schedule III regulations as an anabolic steroid or covered anabolic-steroid substance. Compound-specific human evidence may be limited or historical.

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Anabolic SteroidsModerate class evidence; compound-specific evidence varies

Mesterolone

An orally active DHT-derived androgen used medically in some countries but not broadly approved in the United States. It is androgenic and can suppress endogenous gonadal signaling.

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Anabolic SteroidsSparse/variable compound-specific evidence

Trendione

Trendione is listed in current U.S. federal Schedule III regulations as an anabolic steroid or covered anabolic-steroid substance. Compound-specific human evidence may be limited or historical.

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Anabolic SteroidsModerate class evidence; compound-specific evidence varies

Methandienone

An orally active 17α-alkylated anabolic steroid widely known from historical performance-enhancement use. It is not an FDA-approved dietary supplement and carries the class risks of anabolic-androgenic steroids.

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Anabolic SteroidsSparse/variable compound-specific evidence

13β-Ethyl-17β-hydroxygon-4-en-3-one

13β-Ethyl-17β-hydroxygon-4-en-3-one is listed in current U.S. federal Schedule III regulations as an anabolic steroid or covered anabolic-steroid substance. Compound-specific human evidence may be limited or historical.

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Anabolic SteroidsSparse/variable compound-specific evidence

Methandriol

Methandriol is listed in current U.S. federal Schedule III regulations as an anabolic steroid or covered anabolic-steroid substance. Compound-specific human evidence may be limited or historical.

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Anabolic SteroidsSparse/variable compound-specific evidence

Ethylestrenol

Ethylestrenol is listed in current U.S. federal Schedule III regulations as an anabolic steroid or covered anabolic-steroid substance. Compound-specific human evidence may be limited or historical.

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Anabolic SteroidsModerate class evidence; compound-specific evidence varies

Methasterone

A designer 17α-alkylated anabolic steroid also known as methyldrostanolone or Superdrol. Case literature and class pharmacology raise particular concern for liver and lipid effects.

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Anabolic SteroidsModerate class evidence; compound-specific evidence varies

Fluoxymesterone

A potent 17α-alkylated androgen with historical therapeutic use. Its pharmacology is androgen-receptor mediated; nonmedical exposure can carry substantial hepatic, lipid, cardiovascular and endocrine risk.

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